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Papers authored by Kiselyov AS

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Heterocyclic 1,7-disubstituted indole sulfonamides are potent and selective human EP3 receptor antagonists.

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Hategan G, Polozov AM, Zeller W, Cao H, Mishra RK, Kiselyov AS, Ramirez J, Halldorsdottir G, Andrésson T, Gurney ME, and Singh J

Bioorganic & medicinal chemistry letters 19(23):6797-800, 2009 Dec 1 - Who cited this? | PubMed ID: 19836233 | Fulltext

Synthesis and structural assignment of two major metabolites of the LTA4H inhibitor DG-051.

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Enache LA, Zhang J, Sullins DW, Kennedy I, Onua E, Zembower DE, Muellner FW, Singh J, and Kiselyov AS

Bioorganic & medicinal chemistry letters 19(22):6275-9, 2009 Nov 15 - Who cited this? | PubMed ID: 19819140 | Fulltext

Discovery of leukotriene A4 hydrolase inhibitors using metabolomics biased fragment crystallography.

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Davies DR, Mamat B, Magnusson OT, Christensen J, Haraldsson MH, Mishra R, Pease B, Hansen E, Singh J, Zembower D, Kim H, Kiselyov AS, Burgin AB, Gurney ME, and Stewart LJ

Journal of medicinal chemistry 52(15):4694-715, 2009 Aug 13 - Who cited this? | PubMed ID: 19618939 | Fulltext

(1,2,3-Triazol-4-yl)benzenamines: Synthesis and activity against VEGF receptors 1 and 2.

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Kiselyov AS, Semenova M, and Semenov VV

Bioorganic & medicinal chemistry letters 19(5):1344-8, 2009 Mar 1 - Who cited this? | PubMed ID: 19188066 | Fulltext

3-Acrylamide-4-aryloxyindoles: Synthesis, biological evaluation and metabolic stability of potent and selective EP(3) receptor antagonists.

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Zhou N, Zeller W, Zhang J, Onua E, Kiselyov AS, Ramirez J, Palsdottir G, Halldorsdottir G, Andrésson T, Gurney ME, and Singh J

Bioorganic & medicinal chemistry letters 19(5):1528-31, 2009 Mar 1 - Who cited this? | PubMed ID: 19188065 | Fulltext

3,4-Disubstituted isothiazoles: novel potent inhibitors of VEGF receptors 1 and 2.

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Kiselyov AS, Semenova M, and Semenov VV

Bioorganic & medicinal chemistry letters 19(4):1195-8, 2009 Feb 15 - Who cited this? | PubMed ID: 19124243 | Fulltext

Peri-substituted hexahydro-indolones as novel, potent and selective human EP(3) receptor antagonists.

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O'Connell M, Zeller W, Burgeson J, Mishra RK, Ramirez J, Kiselyov AS, Andrésson T, Gurney ME, and Singh J

Bioorganic & medicinal chemistry letters 19(3):778-82, 2009 Feb 1 - Who cited this? | PubMed ID: 19121942 | Fulltext

Arylphthalazines as potent, and orally bioavailable inhibitors of VEGFR-2.

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Duncton MA, Piatnitski Chekler EL, Katoch-Rouse R, Sherman D, Wong WC, Smith LM, Kawakami JK, Kiselyov AS, Milligan DL, Balagtas C, Hadari YR, Wang Y, Patel SN, Rolster RL, Tonra JR, Surguladze D,

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Bioorganic & medicinal chemistry 17(2):731-40, 2009 Jan 15 - Who cited this? | PubMed ID: 19101155 | Fulltext

3,4-Disubstituted indole acylsulfonamides: a novel series of potent and selective human EP3 receptor antagonists.

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Zhou N, Zeller W, Krohn M, Anderson H, Zhang J, Onua E, Kiselyov AS, Ramirez J, Halldorsdottir G, Andrésson T, Gurney ME, and Singh J

Bioorganic & medicinal chemistry letters 19(1):123-6, 2009 Jan 1 - Who cited this? | PubMed ID: 19022669 | Fulltext

Synthesis and evaluation of heteroaryl-ketone derivatives as a novel class of VEGFR-2 inhibitors.

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Piatnitski Chekler EL, Katoch-Rouse R, Kiselyov AS, Sherman D, Ouyang X, Kim K, Wang Y, Hadari YR, and Doody JF

Bioorganic & medicinal chemistry letters 18(15):4344-7, 2008 Aug 1 - Who cited this? | PubMed ID: 18640036 | Fulltext

Regulators of chemokine receptor activity as promising anticancer therapeutics.

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Balakin KV, Ivanenkov YA, Tkachenko SE, Kiselyov AS, and Ivachtchenko AV

Current cancer drug targets 8(4):299-340, 2008 Jun - Who cited this? | PubMed ID: 18537553 | Fulltext

A synthetic derivative of plant allylpolyalkoxybenzenes induces selective loss of motile cilia in sea urchin embryos.

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Semenova MN, Tsyganov DV, Yakubov AP, Kiselyov AS, and Semenov VV

ACS chemical biology 3(2):95-100, 2008 Feb 15 - Who cited this? | PubMed ID: 18278850 | Fulltext

In vivo Evaluation of Indolyl Glyoxamides in the Phenotypic Sea Urchin Embryo Assay.

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Semenova MN, Kiselyov AS, Titov IY, Raihstat MM, Molodtsov M, Grishchuk E, Spiridonov I, and Semenov VV

Chemical biology & drug design 70(6):485-90, 2007 Dec - Who cited this? | PubMed ID: 17991295 | Fulltext

Novel mitotic targets and their small-molecule inhibitors.

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Ivachtchenko AV, Kiselyov AS, Tkachenko SE, Ivanenkov YA, and Balakin KV

Current cancer drug targets 7(8):766-84, 2007 Dec - Who cited this? | PubMed ID: 18220536 | Fulltext

Histone deacetylase inhibitors in cancer therapy: latest developments, trends and medicinal chemistry perspective.

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Balakin KV, Ivanenkov YA, Kiselyov AS, and Tkachenko SE

Anti-cancer agents in medicinal chemistry 7(5):576-92, 2007 Sep - Who cited this? | PubMed ID: 17896917 | Fulltext

Small-molecule modulators of Hh and Wnt signaling pathways.

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Kiselyov AS, Tkachenko SE, Balakin KV, and Ivachtchenko AV

Expert opinion on therapeutic targets 11(8):1087-101, 2007 Aug - Who cited this? | PubMed ID: 17665980 | Fulltext

Novel inhibitors of VEGF receptors-1 and -2 based on azole-5-carboxamide templates.

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Kiselyov AS, Milligan D, and Ouyang X

Bioorganic & medicinal chemistry letters 17(13):3550-7, 2007 Jul 1 - Who cited this? | PubMed ID: 17481893 | Fulltext

1H-1,2,4-triazol-3-yl-anilines: novel potent inhibitors of vascular endothelial growth factor receptors 1 and 2.

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Kiselyov AS, Piatnitski E, Milligan D, and Ouyang X

Chemical biology & drug design 69(5):331-7, 2007 May - Who cited this? | PubMed ID: 17539825 | Fulltext

ortho-Substituted azoles as selective and dual inhibitors of VEGF receptors 1 and 2.

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Kiselyov AS, Piatnitski EL, Samet AV, Kisliy VP, and Semenov VV

Bioorganic & medicinal chemistry letters 17(5):1369-75, 2007 Mar 1 - Who cited this? | PubMed ID: 17188873 | Fulltext

4-(Azolylphenyl)-phthalazin-1-amines: Novel inhibitors of VEGF receptors I and II.

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Kiselyov AS, Semenov VV, and Milligan D

Chemical biology & drug design 68(6):308-13, 2006 Dec - Who cited this? | PubMed ID: 17177892 | Fulltext

1-(Azolyl)-4-(aryl)-phthalazines: novel potent inhibitors of VEGF receptors I and II.

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Kiselyov AS, Semenova M, Semenov VV, and Piatnitski EL

Chemical biology & drug design 68(5):250-5, 2006 Nov - Who cited this? | PubMed ID: 17177884 | Fulltext

Novel tricyclic azepine derivatives: Biological evaluation of pyrimido[4,5-b]-1,4-benzoxazepines, thiazepines, and diazepines as inhibitors of the epidermal growth factor receptor tyrosine kinase.

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Smith L, Wong WC, Kiselyov AS, Burdzovic-Wizemann S, Mao Y, Xu Y, Duncton MA, Kim K, Piatnitski EL, Doody JF, Wang Y, Rosler RL, Milligan D, Columbus J, Balagtas C, Lee SP,

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Bioorganic & medicinal chemistry letters 16(19):5102-6, 2006 Oct 1 - Who cited this? | PubMed ID: 16887347 | Fulltext

Targeting the hedgehog signaling pathway with small molecules.

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Kiselyov AS

Anti-cancer agents in medicinal chemistry 6(5):445-9, 2006 Sep - Who cited this? | PubMed ID: 17017853 | Fulltext

Natural products as templates for bioactive compound libraries: part 2. Novel modifications of vasicine (peganine) core via efficient and regioselective generation of 3-lithiodeoxyvasicine and its stereoselective addition to aliphatic ketones section sign.

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Shevyakov SV, Davydova OI, Kiselyov AS, Kravchenko DV, Ivachtchenko AV, and Krasavin M

Natural product research 20(9):871-81, 2006 Jul 20 - Who cited this? | PubMed ID: 16753926 | Fulltext

Biology-driven diversity: concept of focused diversity.

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Kiselyov AS

Chemical biology & drug design 68(1):67-9, 2006 Jul - Who cited this? | PubMed ID: 16923028 | Fulltext

Inhibitors of VEGF receptors-1 and -2 based on the 2-((pyridin-4-yl)ethyl)pyridine template.

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Kiselyov AS, Semenova M, Semenov VV, and Milligan D

Bioorganic & medicinal chemistry letters 16(7):1913-9, 2006 Apr 1 - Who cited this? | PubMed ID: 16460936 | Fulltext

Virtual and biomolecular screening converge on a selective agonist for GPR30.

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Bologa CG, Revankar CM, Young SM, Edwards BS, Arterburn JB, Kiselyov AS, Parker MA, Tkachenko SE, Savchuck NP, Sklar LA, Oprea TI, and Prossnitz ER

Nature chemical biology 2(4):207-12, 2006 Apr - Who cited this? | PubMed ID: 16520733 | Fulltext

2-((1H-Azol-1-yl)methyl)-N-arylbenzamides: novel dual inhibitors of VEGFR-1/2 kinases.

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Kiselyov AS, Semenova M, Semenov VV, and Piatnitski E

Bioorganic & medicinal chemistry letters 16(6):1726-30, 2006 Mar 15 - Who cited this? | PubMed ID: 16364640 | Fulltext

Arylphthalazines. Part 2: 1-(Isoquinolin-5-yl)-4-arylamino phthalazines as potent inhibitors of VEGF receptors I and II.

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Duncton MA, Piatnitski EL, Katoch-Rouse R, Smith LM, Kiselyov AS, Milligan DL, Balagtas C, Wong WC, Kawakami J, and Doody JF

Bioorganic & medicinal chemistry letters 16(6):1579-81, 2006 Mar 15 - Who cited this? | PubMed ID: 16386418 | Fulltext

Tricyclic azepine derivatives: pyrimido[4,5-b]-1,4-benzoxazepines as a novel class of epidermal growth factor receptor kinase inhibitors.

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Smith L, Piatnitski EL, Kiselyov AS, Ouyang X, Chen X, Burdzovic-Wizemann S, Xu Y, Pan W, Chen X, Wang Y, Rosler RL, Patel SN, Chiang HH, Milligan DL, Columbus J, Wong WC,

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Bioorganic & medicinal chemistry letters 16(6):1643-6, 2006 Mar 15 - Who cited this? | PubMed ID: 16412636 | Fulltext

Hetaryl imidazoles: a novel dual inhibitors of VEGF receptors I and II.

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Kiselyov AS, Semenova M, Semenov VV, Piatnitski E, and Ouyang S

Bioorganic & medicinal chemistry letters 16(5):1440-4, 2006 Mar 1 - Who cited this? | PubMed ID: 16321531 | Fulltext

Oxadiazole derivatives as a novel class of antimitotic agents: Synthesis, inhibition of tubulin polymerization, and activity in tumor cell lines.

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Ouyang X, Piatnitski EL, Pattaropong V, Chen X, He HY, Kiselyov AS, Velankar A, Kawakami J, Labelle M, Smith L, Lohman J, Lee SP, Malikzay A, Fleming J, Gerlak J, Wang Y,

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Bioorganic & medicinal chemistry letters 16(5):1191-6, 2006 Mar 1 - Who cited this? | PubMed ID: 16377187 | Fulltext

The concept of Focused Diversity: a new algorithm for building screening libraries.

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Kiselyov AS

IDrugs : the investigational drugs journal 9(3):193-8, 2006 Mar - Who cited this? | PubMed ID: 16523385 | Fulltext

Rational design approaches to chemical libraries for hit identification.

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Balakin KV, Kozintsev AV, Kiselyov AS, and Savchuk NP

Current drug discovery technologies 3(1):49-65, 2006 Mar - Who cited this? | PubMed ID: 16712463 | Fulltext

N-(Aryl)-4-(azolylethyl)thiazole-5-carboxamides: novel potent inhibitors of VEGF receptors I and II.

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Kiselyov AS, Piatnitski E, Semenova M, and Semenov VV

Bioorganic & medicinal chemistry letters 16(3):602-6, 2006 Feb - Who cited this? | PubMed ID: 16275072 | Fulltext

N-(4-{[4-(1H-Benzoimidazol-2-yl)-arylamino]-methyl}-phenyl)-benzamide derivatives as small molecule heparanase inhibitors.

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Xu YJ, Miao HQ, Pan W, Navarro EC, Tonra JR, Mitelman S, Camara MM, Deevi DS, Kiselyov AS, Kussie P, Wong WC, and Liu H

Bioorganic & medicinal chemistry letters 16(2):404-8, 2006 Jan 15 - Who cited this? | PubMed ID: 16246551 | Fulltext

1-[4-(1H-Benzoimidazol-2-yl)-phenyl]-3-[4-(1H-benzoimidazol-2-yl)-phenyl]-urea derivatives as small molecule heparanase inhibitors.

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Pan W, Miao HQ, Xu YJ, Navarro EC, Tonra JR, Corcoran E, Lahiji A, Kussie P, Kiselyov AS, Wong WC, and Liu H

Bioorganic & medicinal chemistry letters 16(2):409-12, 2006 Jan 15 - Who cited this? | PubMed ID: 16246560 | Fulltext

Synthesis and structure-activity relationships of 1,2,4-triazoles as a novel class of potent tubulin polymerization inhibitors.

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Ouyang X, Chen X, Piatnitski EL, Kiselyov AS, He HY, Mao Y, Pattaropong V, Yu Y, Kim KH, Kincaid J, Smith L, Wong WC, Lee SP, Milligan DL, Malikzay A, Fleming J,

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Bioorganic & medicinal chemistry letters 15(23):5154-9, 2005 Dec 1 - Who cited this? | PubMed ID: 16198562 | Fulltext

Chemistry of N-fluoropyridinium salts.

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Kiselyov AS

Chemical Society reviews 34(12):1031-7, 2005 Dec - Who cited this? | PubMed ID: 16284669 | Fulltext

Preparation of substituted pyrimido[4,5-b]-1,4-benzoxazepines, thiazepines, and diazepines via a Pictet-Spengler cyclization.

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Duncton MA, Smith LM, Burdzovic-Wizeman S, Burns A, Liu H, Mao Y, Wong WC, and Kiselyov AS

The Journal of organic chemistry 70(23):9629-31, 2005 Nov 11 - Who cited this? | PubMed ID: 16268648 | Fulltext

Arylphthalazines: identification of a new phthalazine chemotype as inhibitors of VEGFR kinase.

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Piatnitski EL, Duncton MA, Kiselyov AS, Katoch-Rouse R, Sherman D, Milligan DL, Balagtas C, Wong WC, Kawakami J, and Doody JF

Bioorganic & medicinal chemistry letters 15(21):4696-8, 2005 Nov 1 - Who cited this? | PubMed ID: 16143524 | Fulltext

Synthesis of polysubstituted 4-fluoroquinolinones.

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Kiselyov AS, Piatnitski EL, and Doody J

Organic letters 6(22):4061-3, 2004 Oct 28 - Who cited this? | PubMed ID: 15496099 | Fulltext

Metabolic activation of benzo[g]chrysene in the human mammary carcinoma cell line MCF-7.

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Agarwal R, Coffing SL, Baird WM, Kiselyov AS, Harvey RG, and Dipple A

Cancer research 57(3):415-9, 1997 Feb 1 - Who cited this? | PubMed ID: 9012467 | Fulltext

Bay-region distortions in a methanol adduct of a bay-region diol epoxide of the carcinogen 5-methylchrysene.

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Afshar CE, Carrell CJ, Carrell HL, Harvey RG, Kiselyov AS, Amin S, and Glusker JP

Carcinogenesis 17(11):2507-11, 1996 Nov - Who cited this? | PubMed ID: 8968070 | Fulltext

Synthesis and structure-DNA binding relationship analysis of DNA triple-helix specific intercalators.

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Strekowski L, Gulevich Y, Baranowski TC, Parker AN, Kiselyov AS, Lin SY, Tanious FA, and Wilson WD

Journal of medicinal chemistry 39(20):3980-3, 1996 Sep 27 - Who cited this? | PubMed ID: 8831763 | Fulltext

Characterization of DNA adducts formed by anti-benzo[g]chrysene 11,12-dihydrodiol 13,14-epoxide.

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Szeliga J, Page JE, Hilton BD, Kiselyov AS, Harvey RG, Dunayevskiy YM, Vouros P, and Dipple A

Chemical research in toxicology 8(8):1014-9, 1995 Dec - Who cited this? | PubMed ID: 8605283 | Fulltext

Mutagenic specificity of syn-benzo[g]chrysene 11,12-dihydrodiol 13,14-epoxide in the dihydrofolate reductase gene of Chinese hamster ovary cells.

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Yuan W, Kiselyov AS, Harvey RG, and Carothers AM

Carcinogenesis 16(11):2869-73, 1995 Nov - Who cited this? | PubMed ID: 7586212 | Fulltext

DNA triple-helix specific intercalators as antigene enhancers: unfused aromatic cations.

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Wilson WD, Tanious FA, Mizan S, Yao S, Kiselyov AS, Zon G, and Strekowski L

Biochemistry 32(40):10614-21, 1993 Oct 12 - Who cited this? | PubMed ID: 8399206 | Fulltext

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