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Papers authored by Bhagwat SS

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AC220 is a uniquely potent and selective inhibitor of FLT3 for the treatment of acute myeloid leukemia (AML).

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Zarrinkar PP, Gunawardane RN, Cramer MD, Gardner MF, Brigham D, Belli B, Karaman MW, Pratz KW, Pallares G, Chao Q, Sprankle KG, Patel HK, Levis M, Armstrong RC, James J, and Bhagwat SS

Blood 114(14):2984-92, 2009 Oct 1 - Who cited this? | PubMed ID: 19654408 | Fulltext

Arylcarboxyamino-substituted diaryl ureas as potent and selective FLT3 inhibitors.

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Patel HK, Grotzfeld RM, Lai AG, Mehta SA, Milanov ZV, Chao Q, Sprankle KG, Carter TA, Velasco AM, Fabian MA, James J, Treiber DK, Lockhart DJ, Zarrinkar PP, and Bhagwat SS

Bioorganic & medicinal chemistry letters 19(17):5182-5, 2009 Sep 1 - Who cited this? | PubMed ID: 19646870 | Fulltext

In Vitro Activity of the Quinolone WCK 771 against Recent U.S. Hospital and Community-Acquired Staphylococcus aureus Pathogens with Various Resistance Types.

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Bhagwat SS, McGhee P, Kosowska-Shick K, Patel MV, and Appelbaum PC

Antimicrobial agents and chemotherapy 53(2):811-3, 2009 Feb - Who cited this? | PubMed ID: 19029326 | Fulltext

Substituted 3-((Z)-2-(4-nitrophenyl)-2-(1H-tetrazol-5-yl) vinyl)-4H-chromen-4-ones as novel anti-MRSA agents: synthesis, SAR, and in-vitro assessment.

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Diwakar SD, Bhagwat SS, Shingare MS, and Gill CH

Bioorganic & medicinal chemistry letters 18(16):4678-81, 2008 Aug 15 - Who cited this? | PubMed ID: 18650090 | Fulltext

Kinase inhibitors for the treatment of inflammatory and autoimmune disorders.

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Bhagwat SS

Purinergic signalling, 2008 Jun 21 - Who cited this? | PubMed ID: 18568424 | Fulltext

4-amino-5-aryl-6-arylethynylpyrimidines: structure-activity relationships of non-nucleoside adenosine kinase inhibitors.

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Matulenko MA, Paight ES, Frey RR, Gomtsyan A, DiDomenico S, Jiang M, Lee CH, Stewart AO, Yu H, Kohlhaas KL, Alexander KM, McGaraughty S, Mikusa J, Marsh KC, Muchmore SW, Jakob CL,

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Bioorganic & medicinal chemistry 15(4):1586-605, 2007 Feb 15 - Who cited this? | PubMed ID: 17197188 | Fulltext

Crystal structures of human adenosine kinase inhibitor complexes reveal two distinct binding modes.

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Muchmore SW, Smith RA, Stewart AO, Cowart MD, Gomtsyan A, Matulenko MA, Yu H, Severin JM, Bhagwat SS, Lee CH, Kowaluk EA, Jarvis MF, and Jakob CL

Journal of medicinal chemistry 49(23):6726-31, 2006 Nov 16 - Who cited this? | PubMed ID: 17154503 | Fulltext

The anti-methicillin-resistant Staphylococcus aureus quinolone WCK 771 has potent activity against sequentially selected mutants, has a narrow mutant selection window against quinolone-resistant Staphylococcus aureus, and preferentially targets DNA gyrase.

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Bhagwat SS, Mundkur LA, Gupte SV, Patel MV, and Khorakiwala HF

Antimicrobial agents and chemotherapy 50(11):3568-79, 2006 Nov - Who cited this? | PubMed ID: 16940059 | Fulltext

Chlorination of aromatic compounds in micellar media: regioselectivity.

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Samant BS, Saraf YP, and Bhagwat SS

Journal of colloid and interface science 302(1):207-13, 2006 Oct 1 - Who cited this? | PubMed ID: 16806254 | Fulltext

Synthesis of new series of 1-Aryl-1,4-dihydro-4-oxo-6-methyl pyridazine-3-carboxylic acid as potential antibacterial agents.

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Nagawade RR, Khanna VV, Bhagwat SS, and Shinde DB

European journal of medicinal chemistry 40(12):1325-30, 2005 Dec - Who cited this? | PubMed ID: 16126308 | Fulltext

Synthesis and biological evaluation of 6,7-disubstituted 4-aminopyrido[2,3-d]pyrimidines as adenosine kinase inhibitors.

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Perner RJ, Lee CH, Jiang M, Gu YG, Didomenico S, Bayburt EK, Alexander KM, Kohlhaas KL, Jarvis MF, Kowaluk EL, and Bhagwat SS

Bioorganic & medicinal chemistry letters 15(11):2803-7, 2005 Jun 2 - Who cited this? | PubMed ID: 15911258 | Fulltext

5-(3-Bromophenyl)-7-(6-morpholin-4-ylpyridin-3-yl)pyrido[2,3-d]pyrimidin-4-ylamine: structure-activity relationships of 7-substituted heteroaryl analogs as non-nucleoside adenosine kinase inhibitors.

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Matulenko MA, Lee CH, Jiang M, Frey RR, Cowart MD, Bayburt EK, Didomenico S, Gfesser GA, Gomtsyan A, Zheng GZ, McKie JA, Stewart AO, Yu H, Kohlhaas KL, Alexander KM, McGaraughty S,

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Bioorganic & medicinal chemistry 13(11):3705-20, 2005 Jun 1 - Who cited this? | PubMed ID: 15863000 | Fulltext

Effect of Lomodex-MgSO(4) in the prevention of reperfusion injury following unilateral testicular torsion: an experimental study in rats.

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Adivarekar PK, Bhagwat SS, Raghavan V, and Bandivdekar AH

Pediatric surgery international 21(3):184-90, 2005 Mar - Who cited this? | PubMed ID: 15711960 | Fulltext

Antistaphylococcal activity of WCK 771, a tricyclic fluoroquinolone, in animal infection models.

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Patel MV, De Souza NJ, Gupte SV, Jafri MA, Bhagwat SS, Chugh Y, Khorakiwala HF, Jacobs MR, and Appelbaum PC

Antimicrobial agents and chemotherapy 48(12):4754-61, 2004 Dec - Who cited this? | PubMed ID: 15561853 | Fulltext

In vitro activity of the new quinolone WCK 771 against staphylococci.

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Jacobs MR, Bajaksouzian S, Windau A, Appelbaum PC, Patel MV, Gupte SV, Bhagwat SS, De Souza NJ, and Khorakiwala HF

Antimicrobial agents and chemotherapy 48(9):3338-42, 2004 Sep - Who cited this? | PubMed ID: 15328094 | Fulltext

Synthesis and biological evaluation of pteridine and pyrazolopyrimidine based adenosine kinase inhibitors.

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Gomtsyan A, Didomenico S, Lee CH, Stewart AO, Bhagwat SS, Kowaluk EA, and Jarvis MF

Bioorganic & medicinal chemistry letters 14(16):4165-8, 2004 Aug 16 - Who cited this? | PubMed ID: 15261263 | Fulltext

Lead identification of a potent benzopyranone selective estrogen receptor modulator.

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McKie JA, Bhagwat SS, Brady H, Doubleday M, Gayo L, Hickman M, Jalluri RK, Khammungkhune S, Kois A, Mortensen D, Richard N, Sapienza J, Shevlin G, Stein B, and Sutherland M

Bioorganic & medicinal chemistry letters 14(13):3407-10, 2004 Jul 5 - Who cited this? | PubMed ID: 15177442 | Fulltext

5,6,7-trisubstituted 4-aminopyrido[2,3-d]pyrimidines as novel inhibitors of adenosine kinase.

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Perner RJ, Gu YG, Lee CH, Bayburt EK, McKie J, Alexander KM, Kohlhaas KL, Wismer CT, Mikusa J, Jarvis MF, Kowaluk EA, and Bhagwat SS

Journal of medicinal chemistry 46(24):5249-57, 2003 Nov 20 - Who cited this? | PubMed ID: 14613327 | Fulltext

Effects of SP500263, a novel selective estrogen receptor modulator, on bone, uterus, and serum cholesterol in the ovariectomized rat.

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Sutherland MK, Brady H, Gayo-Fung LM, Leisten J, Lipps SG, McKie JA, O'Leary E, Patnaik N, Anderson DW, Bhagwat SS, and Stein B

Calcified tissue international 72(6):710-6, 2003 Jun - Who cited this? | PubMed ID: 14563000 | Fulltext

Synthesis and structure-activity relationships of 5-heteroatom-substituted pyridopyrimidines as adenosine kinase inhibitors.

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Gfesser GA, Bayburt EK, Cowart M, DiDomenico S, Gomtsyan A, Lee CH, Stewart AO, Jarvis MF, Kowaluk EA, and Bhagwat SS

European journal of medicinal chemistry 38(3):245-52, 2003 Mar - Who cited this? | PubMed ID: 12667691 | Fulltext

Design, synthesis, and structure-activity relationship of 6-alkynylpyrimidines as potent adenosine kinase inhibitors.

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Gomtsyan A, Didomenico S, Lee CH, Matulenko MA, Kim K, Kowaluk EA, Wismer CT, Mikusa J, Yu H, Kohlhaas K, Jarvis MF, and Bhagwat SS

Journal of medicinal chemistry 45(17):3639-48, 2002 Aug 15 - Who cited this? | PubMed ID: 12166937 | Fulltext

Differential response of estrogen receptors alpha and beta to SP500263, a novel potent selective estrogen receptor modulator.

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Brady H, Doubleday M, Gayo-Fung LM, Hickman M, Khammungkhune S, Kois A, Lipps S, Pierce S, Richard N, Shevlin G, Sutherland MK, Anderson DW, Bhagwat SS, and Stein B

Molecular pharmacology 61(3):562-8, 2002 Mar - Who cited this? | PubMed ID: 11854436 | Fulltext

Effects of SP500263, a novel, potent antiestrogen, on breast cancer cells and in xenograft models.

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Brady H, Desai S, Gayo-Fung LM, Khammungkhune S, McKie JA, O'Leary E, Pascasio L, Sutherland MK, Anderson DW, Bhagwat SS, and Stein B

Cancer research 62(5):1439-42, 2002 Mar 1 - Who cited this? | PubMed ID: 11888917 | Fulltext

SP600125, an anthrapyrazolone inhibitor of Jun N-terminal kinase.

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Bennett BL, Sasaki DT, Murray BW, O'Leary EC, Sakata ST, Xu W, Leisten JC, Motiwala A, Pierce S, Satoh Y, Bhagwat SS, Manning AM, and Anderson DW

Proceedings of the National Academy of Sciences of the United States of America 98(24):13681, 2001 Nov 20 - Who cited this? | PubMed ID: 11717429 | Fulltext

Synthesis and biological evaluation of clitocine analogues as adenosine kinase inhibitors.

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Lee CH, Daanen JF, Jiang M, Yu H, Kohlhaas KL, Alexander K, Jarvis MF, Kowaluk EL, and Bhagwat SS

Bioorganic & medicinal chemistry letters 11(18):2419-22, 2001 Sep 17 - Who cited this? | PubMed ID: 11549437 | Fulltext

Pyridopyrimidine analogues as novel adenosine kinase inhibitors.

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Zheng GZ, Lee C, Pratt JK, Perner RJ, Jiang MQ, Gomtsyan A, Matulenko MA, Mao Y, Koenig JR, Kim KH, Muchmore S, Yu H, Kohlhaas K, Alexander KM, McGaraughty S, Chu KL,

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Bioorganic & medicinal chemistry letters 11(16):2071-4, 2001 Aug 20 - Who cited this? | PubMed ID: 11514141 | Fulltext

Discovery of 4-amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin-3-yl)pyrido[2,3-d]pyrimidine, an orally active, non-nucleoside adenosine kinase inhibitor..

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Lee CH, Jiang M, Cowart M, Gfesser G, Perner R, Kim KH, Gu YG, Williams M, Jarvis MF, Kowaluk EA, Stewart AO, and Bhagwat SS

Journal of medicinal chemistry 44(13):2133-8, 2001 Jun 21 - Who cited this? | PubMed ID: 11405650 | Fulltext

Anti-inflammatory effects of ABT-702, a novel non-nucleoside adenosine kinase inhibitor, in rat adjuvant arthritis.

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Boyle DL, Kowaluk EA, Jarvis MF, Lee CH, Bhagwat SS, Williams M, and Firestein GS

The Journal of pharmacology and experimental therapeutics 296(2):495-500, 2001 Feb - Who cited this? | PubMed ID: 11160636 | Fulltext

Structure-activity studies of 5-substituted pyridopyrimidines as adenosine kinase inhibitors.

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Cowart M, Lee CH, Gfesser GA, Bayburt EK, Bhagwat SS, Stewart AO, Yu H, Kohlhaas KL, McGaraughty S, Wismer CT, Mikusa J, Zhu C, Alexander KM, Jarvis MF, and Kowaluk EA

Bioorganic & medicinal chemistry letters 11(1):83-6, 2001 Jan 8 - Who cited this? | PubMed ID: 11140740 | Fulltext

ABT-702 (4-amino-5-(3-bromophenyl)-7-(6-morpholinopyridin-3-yl)pyrido[2, 3-d]pyrimidine), a novel orally effective adenosine kinase inhibitor with analgesic and anti-inflammatory properties: I. In vitro characterization and acute antinociceptive effects in the mouse.

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Jarvis MF, Yu H, Kohlhaas K, Alexander K, Lee CH, Jiang M, Bhagwat SS, Williams M, and Kowaluk EA

The Journal of pharmacology and experimental therapeutics 295(3):1156-64, 2000 Dec - Who cited this? | PubMed ID: 11082453 | Fulltext

ABT-702 (4-amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin- 3-yl)pyrido[2,3-d]pyrimidine), a novel orally effective adenosine kinase inhibitor with analgesic and anti-inflammatory properties. II. In vivo characterization in the rat.

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Kowaluk EA, Mikusa J, Wismer CT, Zhu CZ, Schweitzer E, Lynch JJ, Lee CH, Jiang M, Bhagwat SS, Gomtsyan A, McKie J, Cox BF, Polakowski J, Reinhart G, Williams M, and Jarvis MF

The Journal of pharmacology and experimental therapeutics 295(3):1165-74, 2000 Dec - Who cited this? | PubMed ID: 11082454 | Fulltext

Adenosine kinase inhibitors.

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Kowaluk EA, Bhagwat SS, and Jarvis MF

Current pharmaceutical design 4(5):403-16, 1998 Oct - Who cited this? | PubMed ID: 10197052 | Fulltext

Isolated jejunal varices.

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Bhagwat SS, Borwankar SS, Ramadwar RH, Naik AS, and Gajaree GI

Journal of postgraduate medicine 41(2):43-4, 1995 - Who cited this? | PubMed ID: 10707708 | Fulltext

Thromboxane receptor antagonism combined with thromboxane synthase inhibition. 5. Synthesis and evaluation of enantiomers of 8-[[(4-chlorophenyl)sulfonyl]amino]-4-(3-pyridinylalkyl)octanoic acid.

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Bhagwat SS, Gude C, Cohen DS, Dotson R, Mathis J, Lee W, and Furness P

Journal of medicinal chemistry 36(2):205-10, 1993 Jan 22 - Who cited this? | PubMed ID: 8423593 | Fulltext

Thromboxane receptor antagonism combined with thromboxane synthase inhibition. 3. Pyridinylalkyl-substituted 8-[(arylsulfonyl)amino]octanoic acids.

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Main AJ, Bhagwat SS, Boswell C, Goldstein R, Gude C, Cohen DS, Furness P, Lee W, and Louzan M

Journal of medicinal chemistry 35(23):4366-72, 1992 Nov 13 - Who cited this? | PubMed ID: 1447737 | Fulltext

Thromboxane receptor antagonism combined with thromboxane synthase inhibition. 4. 8-[[(4-Chlorophenyl)sulfonyl]amino]-4-(3-(3-pyridinyl) propyl)octanoic acid and analogs.

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Bhagwat SS, Gude C, Boswell C, Contardo N, Cohen DS, Dotson R, Mathis J, Lee W, Furness P, and Zoganas H

Journal of medicinal chemistry 35(23):4373-83, 1992 Nov 13 - Who cited this? | PubMed ID: 1447738 | Fulltext

Thromboxane receptor antagonism combined with thromboxane synthase inhibition. 1. (+/-)-(3-pyridinylbicycloheptyl)alkanoic acids.

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Bhagwat SS, Gude C, Cohen DS, Lee W, Furness P, and Clarke FH

Journal of medicinal chemistry 34(6):1790-7, 1991 Jun - Who cited this? | PubMed ID: 1829485 | Fulltext

A study of non-metric (qualitative) variation in Gujarati crania.

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Pal GP, Routal RV, and Bhagwat SS

Anthropologischer Anzeiger; Bericht uber die biologisch-anthropologische Literatur 46(1):65-74, 1988 Mar - Who cited this? | PubMed ID: 3389767 | Fulltext

A study of sutural bones in Gujarati (Indian) crania.

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Pal GP, Bhagwat SS, and Routal RV

Anthropologischer Anzeiger; Bericht uber die biologisch-anthropologische Literatur 44(1):67-76, 1986 Mar - Who cited this? | PubMed ID: 3963790 | Fulltext

Anatomical symmetry in the hind limbs and spinal motoneurons in frogs.

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Pal GP, Routal RV, and Bhagwat SS

Journal of anatomy 143:71-4, 1985 Dec - Who cited this? | PubMed ID: 3870734 | Fulltext

Synthesis and structure of the platelet aggregation factor thromboxane A2.

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Bhagwat SS, Hamann PR, Still WC, Bunting S, and Fitzpatrick FA

Nature 315(6019):511-3, 1985 - Who cited this? | PubMed ID: 4000279 | Fulltext

Observations on brucellosis in Nagpur Region, India.

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Nawathe DR and Bhagwat SS

International journal of zoonoses 11(2):229-32, 1984 Dec - Who cited this? | PubMed ID: 6534910 | Fulltext

The ossification of the membraneous part of the squamous occipital bone in man.

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Pal GP, Tamankar BP, Routal RV, and Bhagwat SS

Journal of anatomy 138 ( Pt 2):259-66, 1984 Mar - Who cited this? | PubMed ID: 6715248 | Fulltext

Melanomas in bullocks.

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Marudwar SS, Bhagwat SS, and Narkhede MD

The Indian veterinary journal 55(8):667-8, 1978 Aug - Who cited this? | PubMed ID: 738792 | Fulltext

Gammaxene poisoning in poultry.

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Bhagwat SS and Jadhav GK

The Indian veterinary journal 45(8):686-8, 1968 Aug - Who cited this? | PubMed ID: 4179661 | Fulltext

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