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Papers authored by Betebenner DA

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Tandem optimization of target activity and elimination of mutagenic potential in a potent series of N-aryl bicyclic hydantoin-based selective androgen receptor modulators.

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Hamann LG, Manfredi MC, Sun C, Krystek SR, Huang Y, Bi Y, Augeri DJ, Wang T, Zou Y, Betebenner DA, Fura A, Seethala R, Golla R, Kuhns JE, Lupisella JA, Darienzo CJ,

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Bioorganic & medicinal chemistry letters 17(7):1860-4, 2007 Apr 1 - Who cited this? | PubMed ID: 17292608 | Fulltext

Inhibitors of HCV NS5B polymerase: synthesis and structure-activity relationships of N-1-benzyl and N-1-[3-methylbutyl]-4-hydroxy-1,8-naphthyridon-3-yl benzothiadiazine analogs containing substituents on the aromatic ring.

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Rockway TW, Zhang R, Liu D, Betebenner DA, McDaniel KF, Pratt JK, Beno D, Montgomery D, Jiang WW, Masse S, Kati WM, Middleton T, Molla A, Maring CJ, and Kempf DJ

Bioorganic & medicinal chemistry letters 16(14):3833-8, 2006 Jul 15 - Who cited this? | PubMed ID: 16650984 | Fulltext

Discovery of a potent inhibitor of the antiapoptotic protein Bcl-xL from NMR and parallel synthesis.

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Petros AM, Dinges J, Augeri DJ, Baumeister SA, Betebenner DA, Bures MG, Elmore SW, Hajduk PJ, Joseph MK, Landis SK, Nettesheim DG, Rosenberg SH, Shen W, Thomas S, Wang X, Zanze I,

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Journal of medicinal chemistry 49(2):656-63, 2006 Jan 26 - Who cited this? | PubMed ID: 16420051 | Fulltext

Discovery and preclinical profile of Saxagliptin (BMS-477118): a highly potent, long-acting, orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes.

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Augeri DJ, Robl JA, Betebenner DA, Magnin DR, Khanna A, Robertson JG, Wang A, Simpkins LM, Taunk P, Huang Q, Han SP, Abboa-Offei B, Cap M, Xin L, Tao L, Tozzo E,

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Journal of medicinal chemistry 48(15):5025-37, 2005 Jul 28 - Who cited this? | PubMed ID: 16033281 | Fulltext

Novel lopinavir analogues incorporating heterocyclic replacements of six-member cyclic urea--synthesis and structure-activity relationships.

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Sham HL, Betebenner DA, Rosenbrook W, Herrin T, Saldivar A, Vasavanonda S, Plattner JJ, and Norbeck DW

Bioorganic & medicinal chemistry letters 14(10):2643-5, 2004 May 17 - Who cited this? | PubMed ID: 15109669 | Fulltext

Synthesis of novel potent dipeptidyl peptidase IV inhibitors with enhanced chemical stability: interplay between the N-terminal amino acid alkyl side chain and the cyclopropyl group of alpha-aminoacyl-l-cis-4,5-methanoprolinenitrile-based inhibitors.

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Magnin DR, Robl JA, Sulsky RB, Augeri DJ, Huang Y, Simpkins LM, Taunk PC, Betebenner DA, Robertson JG, Abboa-Offei BE, Wang A, Cap M, Xin L, Tao L, Sitkoff DF, Malley MF,

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Journal of medicinal chemistry 47(10):2587-98, 2004 May 6 - Who cited this? | PubMed ID: 15115400 | Fulltext

Novel lopinavir analogues incorporating non-Aromatic P-1 side chains--synthesis and structure--activity relationships.

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Sham HL, Zhao C, Li L, Betebenner DA, Saldivar A, Vasavanonda S, Kempf DJ, Plattner JJ, and Norbeck DW

Bioorganic & medicinal chemistry letters 12(21):3101-3, 2002 Nov 4 - Who cited this? | PubMed ID: 12372511 | Fulltext

Synthesis and structure-activity relationships of a novel series of HIV-1 protease inhibitors encompassing ABT-378 (Lopinavir).

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Sham HL, Betebenner DA, Chen X, Saldivar A, Vasavanonda S, Kempf DJ, Plattner JJ, and Norbeck DW

Bioorganic & medicinal chemistry letters 12(8):1185-7, 2002 Apr 22 - Who cited this? | PubMed ID: 11934584 | Fulltext

Synthesis and antiviral activities of the major metabolites of the HIV protease inhibitor ABT-378 (Lopinavir).

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Sham HL, Betebenner DA, Herrin T, Kumar G, Saldivar A, Vasavanonda S, Molla A, Kempf DJ, Plattner JJ, and Norbeck DW

Bioorganic & medicinal chemistry letters 11(11):1351-3, 2001 Jun 4 - Who cited this? | PubMed ID: 11378352 | Fulltext

Novel azacyclic ureas that are potent inhibitors of HIV-1 protease.

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Sham HL, Zhao C, Marsh KC, Betebenner DA, Lin S, Rosenbrook W, Herrin T, Li L, Madigan D, Vasavanonda S, Molla A, Saldivar A, McDonald E, Wideburg NE, Kempf D, Norbeck DW,

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Biochemical and biophysical research communications 225(2):436-40, 1996 Aug 14 - Who cited this? | PubMed ID: 8753780 | Fulltext

A novel, picomolar inhibitor of human immunodeficiency virus type 1 protease.

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Sham HL, Zhao C, Stewart KD, Betebenner DA, Lin S, Park CH, Kong XP, Rosenbrook W, Herrin T, Madigan D, Vasavanonda S, Lyons N, Molla A, Saldivar A, Marsh KC, McDonald E,

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Journal of medicinal chemistry 39(2):392-7, 1996 Jan 19 - Who cited this? | PubMed ID: 8558507 | Fulltext

Potent inhibitors of the HIV-1 protease with good oral bioavailabilities.

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Sham HL, Zhao C, Marsh KC, Betebenner DA, Lin S, McDonald E, Vasavanonda S, Wideburg N, Saldivar A, and Robins T

Biochemical and biophysical research communications 211(1):159-65, 1995 Jun 6 - Who cited this? | PubMed ID: 7779082 | Fulltext

Pseudo-symmetrical difluoroketones. Highly potent and specific inhibitors of HIV-1 protease.

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Sham HL, Betebenner DA, Wideburg N, Saldivar AC, Kohlbrenner WE, Craig-Kennard A, Vasavanonda S, Kempf DJ, Clement JJ, and Erickson JE

FEBS letters 329(1-2):144-6, 1993 Aug 23 - Who cited this? | PubMed ID: 8354389 | Fulltext

Potent HIV-1 protease inhibitors with antiviral activities in vitro.

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Sham HL, Betebenner DA, Wideburg NE, Saldivar AC, Kohlbrenner WE, Vasavanonda S, Kempf DJ, Norbeck DW, Zhao C, and Clement JJ

Biochemical and biophysical research communications 175(3):914-9, 1991 Mar 29 - Who cited this? | PubMed ID: 2025263 | Fulltext

Hepatobiliary delivery of polyaminopolycarboxylate chelates: synthesis and characterization of a cholic acid conjugate of EDTA and biodistribution and imaging studies with its indium-111 chelate.

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Betebenner DA, Carney PL, Zimmer AM, Kazikiewicz JM, Brücher E, Sherry AD, and Johnson DK

Bioconjugate chemistry 2(2):117-23, 1991 - Who cited this? | PubMed ID: 1907855 | Fulltext

Carboxymethyl-substituted bifunctional chelators: preparation of aryl isothiocyanate derivatives of 3-(carboxymethyl)-3-azapentanedioic acid, 3,12-bis(carboxymethyl)-6,9-dioxa-3,12-diazatetradecanedioic++ + acid, and 1,4,7,10-tetraazacyclododecane-N,N',N",N'''-tetraacetic acid for use as protein labels.

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Kline SJ, Betebenner DA, and Johnson DK

Bioconjugate chemistry 2(1):26-31, 1991 - Who cited this? | PubMed ID: 1908704 | Fulltext

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