Papers authored by Augeri DJ

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5-Fluorocytosine derivatives as inhibitors of deoxycytidine kinase.
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Tarver JE, Jessop TC, Carlsen M, Augeri DJ, Fu Q, Healy JP, Heim-Riether A, Xu A, Taylor JA, Shen M, Keyes PE, David Kimball S, Yu XC, Miranda M, Liu Q, Swaffield JC, 
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Bioorganic & medicinal chemistry letters 19(23):6780-3, 2009 Dec 1 - Who cited this? | PubMed ID: 19836229 | Fulltext
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Lead optimization and structure-based design of potent and bioavailable deoxycytidine kinase inhibitors.
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Jessop TC, Tarver JE, Carlsen M, Xu A, Healy JP, Heim-Riether A, Fu Q, Taylor JA, Augeri DJ, Shen M, Stouch TR, Swanson RV, Tari LW, Hunter M, Hoffman I, Keyes PE, 
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Bioorganic & medicinal chemistry letters 19(23):6784-7, 2009 Dec 1 - Who cited this? | PubMed ID: 19836232 | Fulltext
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Inhibition of sphingosine-1-phosphate lyase for the treatment of autoimmune disorders.
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Bagdanoff JT, Donoviel MS, Nouraldeen A, Tarver J, Fu Q, Carlsen M, Jessop TC, Zhang H, Hazelwood J, Nguyen H, Baugh SD, Gardyan M, Terranova KM, Barbosa J, Yan J, Bednarz M, 
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Journal of medicinal chemistry 52(13):3941-53, 2009 Jul 9 - Who cited this? | PubMed ID: 19489538 | Fulltext
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Potent non-nitrile dipeptidic dipeptidyl peptidase IV inhibitors.
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Simpkins LM, Bolton S, Pi Z, Sutton JC, Kwon C, Zhao G, Magnin DR, Augeri DJ, Gungor T, Rotella DP, Sun Z, Liu Y, Slusarchyk WS, Marcinkeviciene J, Robertson JG, Wang A, 
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Bioorganic & medicinal chemistry letters 17(23):6476-80, 2007 Dec 1 - Who cited this? | PubMed ID: 17937986 | Fulltext
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Tandem optimization of target activity and elimination of mutagenic potential in a potent series of N-aryl bicyclic hydantoin-based selective androgen receptor modulators.
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Hamann LG, Manfredi MC, Sun C, Krystek SR, Huang Y, Bi Y, Augeri DJ, Wang T, Zou Y, Betebenner DA, Fura A, Seethala R, Golla R, Kuhns JE, Lupisella JA, Darienzo CJ, 
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Bioorganic & medicinal chemistry letters 17(7):1860-4, 2007 Apr 1 - Who cited this? | PubMed ID: 17292608 | Fulltext
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Discovery of a potent inhibitor of the antiapoptotic protein Bcl-xL from NMR and parallel synthesis.
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Petros AM, Dinges J, Augeri DJ, Baumeister SA, Betebenner DA, Bures MG, Elmore SW, Hajduk PJ, Joseph MK, Landis SK, Nettesheim DG, Rosenberg SH, Shen W, Thomas S, Wang X, Zanze I, 
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Journal of medicinal chemistry 49(2):656-63, 2006 Jan 26 - Who cited this? | PubMed ID: 16420051 | Fulltext
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Discovery and preclinical profile of Saxagliptin (BMS-477118): a highly potent, long-acting, orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes.
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Augeri DJ, Robl JA, Betebenner DA, Magnin DR, Khanna A, Robertson JG, Wang A, Simpkins LM, Taunk P, Huang Q, Han SP, Abboa-Offei B, Cap M, Xin L, Tao L, Tozzo E, 
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Journal of medicinal chemistry 48(15):5025-37, 2005 Jul 28 - Who cited this? | PubMed ID: 16033281 | Fulltext
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An inhibitor of Bcl-2 family proteins induces regression of solid tumours.
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Oltersdorf T, Elmore SW, Shoemaker AR, Armstrong RC, Augeri DJ, Belli BA, Bruncko M, Deckwerth TL, Dinges J, Hajduk PJ, Joseph MK, Kitada S, Korsmeyer SJ, Kunzer AR, Letai A, Li C, 
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Nature 435(7042):677-81, 2005 Jun 2 - Who cited this? | PubMed ID: 15902208 | Fulltext
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Synthesis of novel potent dipeptidyl peptidase IV inhibitors with enhanced chemical stability: interplay between the N-terminal amino acid alkyl side chain and the cyclopropyl group of alpha-aminoacyl-l-cis-4,5-methanoprolinenitrile-based inhibitors.
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Magnin DR, Robl JA, Sulsky RB, Augeri DJ, Huang Y, Simpkins LM, Taunk PC, Betebenner DA, Robertson JG, Abboa-Offei BE, Wang A, Cap M, Xin L, Tao L, Sitkoff DF, Malley MF, 
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Journal of medicinal chemistry 47(10):2587-98, 2004 May 6 - Who cited this? | PubMed ID: 15115400 | Fulltext
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NMR-based modification of matrix metalloproteinase inhibitors with improved bioavailability.
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Hajduk PJ, Shuker SB, Nettesheim DG, Craig R, Augeri DJ, Betebenner D, Albert DH, Guo Y, Meadows RP, Xu L, Michaelides M, Davidsen SK, and Fesik SW
Journal of medicinal chemistry 45(26):5628-39, 2002 Dec 19 - Who cited this? | PubMed ID: 12477346 | Fulltext
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Novel inhibitors of Erm methyltransferases from NMR and parallel synthesis.
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Hajduk PJ, Dinges J, Schkeryantz JM, Janowick D, Kaminski M, Tufano M, Augeri DJ, Petros A, Nienaber V, Zhong P, Hammond R, Coen M, Beutel B, Katz L, and Fesik SW
Journal of medicinal chemistry 42(19):3852-9, 1999 Sep 23 - Who cited this? | PubMed ID: 10508434 | Fulltext
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Potent and orally bioavailable noncysteine-containing inhibitors of protein farnesyltransferase.
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Augeri DJ, Janowick D, Kalvin D, Sullivan G, Larsen J, Dickman D, Ding H, Cohen J, Lee J, Warner R, Kovar P, Cherian S, Saeed B, Zhang H, Tahir S, Ng SC, 
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Bioorganic & medicinal chemistry letters 9(8):1069-74, 1999 Apr 19 - Who cited this? | PubMed ID: 10328287 | Fulltext
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Potent and selective non-cysteine-containing inhibitors of protein farnesyltransferase.
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Augeri DJ, O'Connor SJ, Janowick D, Szczepankiewicz B, Sullivan G, Larsen J, Kalvin D, Cohen J, Devine E, Zhang H, Cherian S, Saeed B, Ng SC, and Rosenberg S
Journal of medicinal chemistry 41(22):4288-300, 1998 Oct 22 - Who cited this? | PubMed ID: 9784104 | Fulltext
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